Itekhnoloji yeGlycopeptide

Ngokwendlela yokudibanisa ye-amino acid kunye noshukela, i-peptide yeswekile inokwahlulwa ibe ngamacandelo amane: i-O glycosylation, i-C a N glycosylation, i-saccharification yamazolo kunye ne-GPI (glycophosphatidlyinositol) uxhumano.

1. I-N-glycosylation glycopeptides yenziwe nge-N-acetamide i-glucose ekupheleni kokunciphisa i-glycan chain (i-Glc-Nac) edityaniswe ne-athomu ye-N kwiqela le-amide yecala lecala le-Asn kwi-peptide chain, kunye ne-Asn. ekwazi ukudibanisa ikhonkco ye-glycan kufuneka ibekwe kwi-AsN-X-Ser / Thr (X! = P) kwi-motif eyenziwe ngama-residu.Iswekile yiN-acetylglucosamine.

N-糖基化修饰结构糖肽

I-N-glycosylation eguqulelwe kwi-structural glycopeptide

2. Isakhiwo se-O-glycosylation silula kune-N-glycosylation.Le glycopeptide imfutshane ngokubanzi kune-glycan, kodwa ineentlobo ezininzi kune-N-glycosylation.I-Ser kunye ne-Thr ngokubanzi zinokufakwa kwi-glycosylated kwikhonkco le-peptide.Ukongeza, kukho i-glycopeptides ehonjiswe nge-tyrosine, i-hydroxyl, kunye ne-hydroxyproline glycosylation.Indawo yekhonkco yi-athomu ye-oksijini ye-hydroxyl kwicala lekhonkco lentsalela.Iishukela ezidibeneyo ziyi-galactose okanye i-N-acetylgalactosamine (i-Gal & GalNAc) okanye i-glucose / glucosamine (Glc / GlcNAc), i-mannose / mannosamine (Man / ManNAc), njl.

O-糖基化修饰结构

I-O-glycosylation iguqula isakhiwo

3. I-Glycopeptide O-GlcNAC glycosylation ((N-acetylcysteine ​​(NAC)) (glcnAcN-acetylglucosamine/acetylglucosamine)

I-N-acetylglucosamine enye (GlcNAc) i-glycosylation idibanisa iiprotheni ze-O-GlcNAc kwi-athomu ye-oksijini ye-hydroxyl ye-serine okanye i-threonine intsalela yeprotheni.I-O-GlcNA glycosylation yi-O-GlcNAc monosaccharide ihombiso ngaphandle kokwandiswa kwe-glycan;Njenge-peptide phosphorylation, i-O-GlcNAc glycosylation ye-glycopeptides ikwayinkqubo yokuhombisa iprotein eguqukayo.Ukuhonjiswa okungaqhelekanga kwe-O-GlcNAc kunokubangela izifo ezahlukeneyo ezifana nesifo seswekile, izifo zentliziyo, ithumba, isifo sika-Alzheimer njalo njalo.

Amanqaku e-glycosylation ye-glycopeptides

Izakhiwo ezisisiseko ze-polypeptide kunye ne-sugar chain zidibaniswe namatyathanga eprotheyini ngamabhondi adibeneyo, kwaye iziza ezidibanisa amatyathanga eswekile zibizwa ngokuba ziindawo ze-glycosylation.Ekubeni akukho template yokulandela i-biosynthesis ye-glycopeptide sugar chain, i-sugar chain ezahlukeneyo ziya kuqhotyoshelwa kwindawo efanayo ye-glycosylation, ekhokelela kwinto ebizwa ngokuba yi-microscopic inhomogeneity.

I-glycosylation ye-glycopeptides

1. Impembelelo ye-glycopeptide glycosylation kunyango-impumelelo yeeproteni zonyango.

Kwimeko yeeprotheyini zonyango-zonyango, i-glycosylation ikwachaphazela isiqingatha sobomi kunye nokujoliswa kweziyobisi zeprotheyini kwi-vivo.

2. I-glycopeptide e-Soluble glycosylation kunye neeprotheni

Uphononongo lubonise ukuba amatyathanga eswekile kumphezulu weeproteni anokuphucula ukunyibilika kwemolekyuli yeeproteni

3. I-Glycopeptide glycosylation kunye ne-protein immunogenicity

Kwelinye icala, amatyathanga eswekile kumphezulu weeproteni anokubangela iimpendulo ezithile zokuzikhusela kwizifo.Kwelinye icala, amatyathanga eswekile anokugquma iindawo ezithile kumphezulu weprotein kwaye anciphise ukungazinzi kwawo

4. I-Glycopeptide glycosylation eyandisa ukuzinza kweprotheni

I-Glycosylation inokunyusa ukuzinza kweeprotheni kwiimeko ezahlukeneyo ze-denaturation (ezifana ne-denaturants, ukushisa, njl.) kwaye ugweme ukuhlanganiswa kweeprotheni.Kwangaxeshanye, imixokelelwane yeswekile kumphezulu weeproteni inokugquma iindawo zokuwohloka kweproteolytic yeemolekyuli zeprotheyini, ngaloo ndlela inyusa ukuxhathisa kweeprotheyini kwiiprotheyini.

5. I-Glycopeptide glycosylation echaphazela umsebenzi webhayoloji weemolekyuli zeprotheni

Ukutshintsha iprotein glycosylation kunokwenza ukuba iimolekyuli zeprotheyini zenze imisebenzi emitsha yebhayoloji


Ixesha lokuposa: Aug-03-2023